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VSV

Indiana vesiculovirus

4
Approved Drugs
0
Phase 3
0
Phase 2
16
Preclinical
20
Total Compounds

Antiviral Compounds

AmantadineVSVViroporin inhibitor; blocks viral ion channel activity
Approved (other)
Japan
Viral ion channel (viroporin)
AmiodaroneVSVNon-competitive β-adrenergic inhibitor
Preclinical
—Human (multiple)
AmodiaquineVSVMethyltransferase inhibitor
Preclinical
—Human HNMT
BortezomibVSVProteasome inhibitor (26S subunit)
Preclinical
—Human proteasome
BrequinarVSVDHODH (DHODH) inhibitor
Preclinical
—Human DHODH
ClotrimazoleVSVBlock Viral Entry (KCa3.1 antagonist)
Preclinical
—Human cytochrome P450
CyclosporineVSVCalcineurin inhibitor; allows for inhibition of T cell activation
Preclinical
—Human CYPs
DoxycyclineVSV—
Preclinical
—Unknown
EflornithineVSVEnzyme-activated; irreversible inhibitor of ornithine decarboxylase
Preclinical
—Human ODC
FoscarnetVSVPyrophosphate analog DNA polymerase inhibitor
Approved (other)
Japan
Viral RNA pol
IndomethacinVSVCyclo-oxygenase (COX) enzyme or prostaglandin G/H synthase inhibitor
Preclinical
—Human COX
JIB-04VSVHuman HDAC inhibitor
Preclinical
—Human HDAC
MonensinVSV—
Preclinical
—Unknown
NelfinavirVSVHIV protease inhibitor
Approved (other)
Japan
Unknown
NiclosamideVSV—
Preclinical
—Human (multiple)
PodofiloxVSV—
Preclinical
—Human topoisomerase
RaloxifeneVSVSelective estrogen receptor modulator
Preclinical
—Human (multiple)
RegorafenibVSVB-Raf; c-Kit; VEGFR2 inhibitor
Preclinical
—Human PTK
SaquinavirVSVProtease inhibitor
Approved (other)
JapanRussia
Unknown
SorafenibVSVB-Raf; FGFR-1; VEGFR-2 & -3; PDGFR-beta; KIT; and FLT3 inhibitor
Preclinical
—Human PTK
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