Human immunodeficiency virus (HIV)
| Zidovudine | HIV | — | FDA approved | FDAJapanRussia | NRTIs | AntiviralDbpmda.go.jp |
| Didanosine | HIV | — | FDA approved | FDAJapan | NRTIs | AntiviralDbpmda.go.jp |
| Zalcitabine | HIV | — | FDA approved | FDAJapan | NRTIs | AntiviralDbpmda.go.jp |
| Stavudine | HIV | — | FDA approved | FDAJapanRussia | NRTIs | AntiviralDbpmda.go.jp |
| Lamivudine | HIV | — | FDA approved | FDAJapanChinaRussia | NRTIs | |
| Abacavir | HIV | — | FDA approved | FDAJapanRussia | NRTIs | AntiviralDbpmda.go.jp |
| Emtricitabine | HIV | — | FDA approved | FDAJapanRussia | NRTIs | |
| Tenofovir alafenamide | HIV | — | FDA approved | FDAJapanChina | NRTIs | |
| Nevirapine | HIV | — | FDA approved | FDAJapanRussia | NNRTIs | AntiviralDbpmda.go.jp |
| Delavirdine | HIV | — | FDA approved | FDAJapan | NNRTIs | |
| Efavirenz | HIV | — | FDA approved | FDAJapanRussia | NNRTIs | AntiviralDbpmda.go.jp |
| Elsulfavirine | HIV | — | Approved (other) | Russia | NNRTIs | AntiviralDb |
| Etravirine | HIV | — | FDA approved | FDAJapan | NNRTIs | |
| Rilpivirine | HIV | — | FDA approved | FDAJapan | NNRTIs | |
| Doravirine | HIV | — | FDA approved | FDAJapan | NNRTIs | |
| Saquinavir | HIV | — | FDA approved | FDAJapanRussia | Protease | AntiviralDbpmda.go.jp |
| Indinavir | HIV | — | FDA approved | FDAJapan | Protease | AntiviralDbpmda.go.jp |
| Amprenavir | HIV | — | FDA approved | FDAJapan | Protease | AntiviralDbpmda.go.jp |
| Atazanavir | HIV | — | FDA approved | FDAJapanRussia | Protease | |
| Fosamprenavir | HIV | — | FDA approved | FDAJapan | Protease | |
| Tipranavir | HIV | — | FDA approved | FDA | Protease | AntiviralDb |
| Darunavir | HIV | — | FDA approved | FDAJapanRussia | Protease | |
| Raltegravir | HIV | — | FDA approved | FDAJapan | Integrase | |
| Elvitegravir | HIV | — | FDA approved | FDAJapan | Integrase | |
| Dolutegravir | HIV | — | FDA approved | FDAJapan | Integrase |