Retroviridae · Lentivirus
| Lopinavir | HIV-2 | HIV protease inhibitor | FDA approved | FDAJapanRussia | Viral protease | |
| Ritonavir | HIV-2 | HIV protease inhibitor | FDA approved | FDAJapanRussia | Viral protease | |
| Tenofovir | HIV-2 | Nucleotide analog RT inhibitor | FDA approved | FDAChinaRussia | Viral RT | |
| Azacitidine | HIV-2 | Nucleoside analog DNA methyl transferase inhibitor | Preclinical | — | Viral RT | |
| Cenicriviroc | HIV-2 | Unknown | Preclinical | — | Human CCR5 | |
| Lamivudine | HIV-2 | RT inhibitor and zalcitabine analog | FDA approved | FDAJapanChinaRussia | Viral RT |